Table1: HDACIs and their involvements in myocardial
infarction.
HDACIs |
Targets |
Function
|
Signaling
pathway Reference |
VPA |
Increase t-PA release |
Improve endogenous fibrinolytic capacity; reduced risk for myocardial
infarction |
|
CPA |
Inhibit HDAC2 |
Prevent neointima
formation, adipocytic differentiation, lipid
accumulation |
|
SAHA |
Inhibit HDAC1,2 |
Reduce infarct size; promote
autophagy |
|
TSA |
Inhibit HDAC1,2 |
Stimulates myogenesis
and angiogenesis; reduce infarct size |
|
Scipataid Mocetinostat |
Synthetic HDACI Inhibit HDAC 1,2,3 |
Reduce infarct size |